Synthesis and Chemistry of Agrochemicals III

by Baker, Don R.; Fenyes, Joseph G.; Steffens, James J.

• ISBN13: 9780841224735
• ISBN10: 0841224730
• Format: Hardcover
• Copyright: 1992-05-05
• Publisher: American Chemical Society

Summary

Covers the discovery, development, and optimization of new agrochemicals. Discusses new structures, new synthesis strategies, and structure-activity relationships of agrochemicals for plant control; insect, acarid, and nematode control; and fungal disease control. Also examines many of the toxicological problems encountered during development of new agrochemicals. Case histories describe the discovery and development of specific agrochemicals. Presents material and information that previously has only partially appeared in the patent literature.

Table of Contents

Progress in a Time of Change1,2,4-Triazolo[1,5-a]pyrimidine-2-sulfonanilide Herbicides: Influence of Alkyl,Haloalkyl, and Halogen Heterocyclic Substitution on In Vitro and In Vivo

Biological Activity1,2,4-Triazolo[1,5-a]pyrimidine-2-sulfonanilide Herbicides: Influence of Alkoxy

Heterocyclic Substitution on In Vitro and In Vivo Biological Activity and Soil

DecompositionN-(Substituted-2-fluorophenyl)- and N-(Substituted-2-trifluormethylphenyl)-1,2,4-triazolo -[1,5-a]pyrimidine-2-sulfonanilides:Synthesis and Herbicidal Activity

New Pyrazole Sulfonylureas: Synthesis and Herbicidal Activity

Synthesis and Quantitative Structure-Activity Relationships of

Pyridylsulfonylurea Herbicides

Novel N-Substituted Imidazolinones: Synthesis and Herbicidal Activity

Discovery of a New Class of Herbicides: Sulfonyl Carboxamides

Phenyl-Substituted Five-Membered-Ring Heterocycles as Bleaching Herbicides7-Phenyl-1,2,4-triazolo[1,5-a]pyrimidines and Related Heterocycles: A New Familyof Bleaching Herbicides

Diphenylpyridines: A New Class of Herbicides

Structure-Activity Relationships in 3-Alkyl- and 3-Aryl-5-isothiazolylureas:Pre- and Postemergence Herbicides with Two Possible Modes of Action

Design and Synthesis of 1-Aryl-4-substituted-1,4-dihydro-5H-tetrazol-5-ones: ANovel Pre- and Postemergence Class of Herbicides

Synthesis and Herbicidal Properties of Aryltriazolinones: A New Class of Pre-and Postemergence Herbicides

Novel Pryazole Phenyl Ether Herbidices

N-Substituted-2,6-(polyfluoromethyl)dihydropyridine-3,5- dicarboxylates:Synthesis and Herbicidal Activity5-Substituted-2,4-imidazolidinediones: Synthesis and Herbicidal Activity

Cyanoacrylate Inhibitors of Photosynthetic Electron Transport: Structural

Requirements for Inhibitor Potency and Herbicidal Activity

Synthesis and Gametocidal Activity of1-Aryl-5-(aminocarbonyl)-1H-pyrazole-4-carboxylic Acids

Discovery, Isolation, and Structure Elucidation of a Family of Structurally

Unique, Fermentation-Derived Tetracyclic Macrolides

New Series of Milbemycin Macrolides (LL-F28249) with Endectocidal, Insecticidal,and Acaricidal Activity: Synthetic Modification and Biological Activity

Regio- and Stereoselective Synthesis of 13b-Substituted-milbemycins, includingthe 13b-Alkyl-milbemycins

Highly Efficacious Non-Ester Pyrethroid Insecticides with Low Toxicity to Fish1,4-Diaryl-1-cyclopropylbutanes: Highly Efficacious Insecticides with Low Fish

Toxicity

Insecticidal Pyrroles: Discovery and Overview

Insecticidal Pyrroles: Arylpyrrolecarbonitriles Incorporating a Trifluoromethyl

Group

Insecticidal Pyrroles: Synthesis of bis-(Trifluoromethyl) Pyrroles via

Rearrangement of O-Vinyloximes

Insecticidal Dihydropyrazoles with Reduced Lipophilicity

N-Benzoyl-N-alkyl-2-aminothiazole Proinsecticides

Diphenylamines I: Synthesis and Structure-Activity Relationship Development of

Novel N-(Substituted Phenyl)-N-alkyl-2-(trifluoromethyl)-4,6-dinitrobenzenamines

Leading to a Potent Miticide(EL-462)Diphenylamines II: Synthesis and Miticidal Activity of 2-Alkyl-4,6-dinitro- and4-Alkyl-2,6-dinitrodiphenylamine Analogs and Derivatives

Synthesis and Reactivity of Cyclic Hydroxamic Acids: Resistance Factors in the

Gramineae

Nematicidal Activity of5-Substituted-2-S-(3,4,4-trifluoro-3-butenyl)-1,3,4-thiadiazoles

Fungicidal b-Methoxyacrylates: From Natural Products to Novel Synthetic

Agricultural Fungicides

Total Synthesis of Naturally Occurring 1,2-Dithiolo[4,3-b]pyrrolones and Related

Compounds

Phenylpyrroles, a New Class of Agricultural Fungicides Related to the Natural

Antibiotic Pyrrolnitrin

Synthesis of Fungicidal Phenylpyrroles

Design of Sterol Reductase Inhibitors: Insights into the Binding Conformation of

Tertiary Amine Fungicides

Mechanism of the Antifungal Action of (S)-2-Amino-4-oxo-5-hydroxypentanoic Acid,RI-331: Inhibition of Homoserine Dehydrogenase in Saccharomyces cerevisiae

A Novel Class of Benzamide Fungicides

Table of Contents provided by Publisher. All Rights Reserved.